Synthesis of DNA-Sequence-Selective Hairpin Polyamide Platinum Complexes

Two DNA-sequence-selective hairpin polyamide platinum(II) complexes, containing pyrrole and imidazole heterocyclic rings, have been synthesised by different methods. A six-ring complex, selective for (A/T)GGG(A/T) DNA sequences, was made by using solid-phase synthesis, whilst an eight-ring complex,...

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محفوظ في:
التفاصيل البيبلوغرافية
المؤلف الرئيسي: Taleb, Robin (author)
مؤلفون آخرون: Jaramillo, David (author), Wheate, Nial (author), Aldrich-Wright, Janice (author)
التنسيق: article
منشور في: 2007
الوصول للمادة أونلاين:http://hdl.handle.net/10725/3496
http://dx.doi.org/10.1002/chem.200601486
http://onlinelibrary.wiley.com/doi/10.1002/chem.200601486/full
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author Taleb, Robin
author2 Jaramillo, David
Wheate, Nial
Aldrich-Wright, Janice
author2_role author
author
author
author_facet Taleb, Robin
Jaramillo, David
Wheate, Nial
Aldrich-Wright, Janice
author_role author
dc.creator.none.fl_str_mv Taleb, Robin
Jaramillo, David
Wheate, Nial
Aldrich-Wright, Janice
dc.date.none.fl_str_mv 2007
2016-04-06T05:57:47Z
2016-04-06T05:57:47Z
2016-04-06
dc.identifier.none.fl_str_mv 0947-6539
http://hdl.handle.net/10725/3496
http://dx.doi.org/10.1002/chem.200601486
Taleb, R. I., Jaramillo, D., Wheate, N. J., & Aldrich‐Wright, J. R. (2007). Synthesis of DNA‐Sequence‐Selective Hairpin Polyamide Platinum Complexes. Chemistry–A European Journal, 13(11), 3177-3186.
http://onlinelibrary.wiley.com/doi/10.1002/chem.200601486/full
dc.language.none.fl_str_mv en
dc.relation.none.fl_str_mv Chemistry a European Journal
dc.rights.*.fl_str_mv info:eu-repo/semantics/openAccess
dc.title.none.fl_str_mv Synthesis of DNA-Sequence-Selective Hairpin Polyamide Platinum Complexes
dc.type.none.fl_str_mv Article
info:eu-repo/semantics/publishedVersion
info:eu-repo/semantics/article
description Two DNA-sequence-selective hairpin polyamide platinum(II) complexes, containing pyrrole and imidazole heterocyclic rings, have been synthesised by different methods. A six-ring complex, selective for (A/T)GGG(A/T) DNA sequences, was made by using solid-phase synthesis, whilst an eight-ring complex, selective for (A/T)CCTG(A/T) DNA sequences, was made by utilising standard wet chemistry. Solid-phase synthesis resulted in a significantly higher yield, required less purification and is more efficient than the wet synthesis; as such, it is the preferred method for further work. The metal complexes were characterised by 1H and 195Pt NMR spectroscopy and ESI mass spectrometry. The two compounds provide a foundation for the synthesis of more complex molecules containing multiple hairpins and/or platinum groups.
eu_rights_str_mv openAccess
format article
id LAURepo_befaa33a2176c061548a564b70679fa0
identifier_str_mv 0947-6539
Taleb, R. I., Jaramillo, D., Wheate, N. J., & Aldrich‐Wright, J. R. (2007). Synthesis of DNA‐Sequence‐Selective Hairpin Polyamide Platinum Complexes. Chemistry–A European Journal, 13(11), 3177-3186.
language_invalid_str_mv en
network_acronym_str LAURepo
network_name_str Lebanese American University repository
oai_identifier_str oai:laur.lau.edu.lb:10725/3496
publishDate 2007
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spelling Synthesis of DNA-Sequence-Selective Hairpin Polyamide Platinum ComplexesTaleb, RobinJaramillo, DavidWheate, NialAldrich-Wright, JaniceTwo DNA-sequence-selective hairpin polyamide platinum(II) complexes, containing pyrrole and imidazole heterocyclic rings, have been synthesised by different methods. A six-ring complex, selective for (A/T)GGG(A/T) DNA sequences, was made by using solid-phase synthesis, whilst an eight-ring complex, selective for (A/T)CCTG(A/T) DNA sequences, was made by utilising standard wet chemistry. Solid-phase synthesis resulted in a significantly higher yield, required less purification and is more efficient than the wet synthesis; as such, it is the preferred method for further work. The metal complexes were characterised by 1H and 195Pt NMR spectroscopy and ESI mass spectrometry. The two compounds provide a foundation for the synthesis of more complex molecules containing multiple hairpins and/or platinum groups.PublishedN/A2016-04-06T05:57:47Z2016-04-06T05:57:47Z20072016-04-06Articleinfo:eu-repo/semantics/publishedVersioninfo:eu-repo/semantics/article0947-6539http://hdl.handle.net/10725/3496http://dx.doi.org/10.1002/chem.200601486Taleb, R. I., Jaramillo, D., Wheate, N. J., & Aldrich‐Wright, J. R. (2007). Synthesis of DNA‐Sequence‐Selective Hairpin Polyamide Platinum Complexes. Chemistry–A European Journal, 13(11), 3177-3186.http://onlinelibrary.wiley.com/doi/10.1002/chem.200601486/fullenChemistry a European Journalinfo:eu-repo/semantics/openAccessoai:laur.lau.edu.lb:10725/34962016-08-12T09:28:59Z
spellingShingle Synthesis of DNA-Sequence-Selective Hairpin Polyamide Platinum Complexes
Taleb, Robin
status_str publishedVersion
title Synthesis of DNA-Sequence-Selective Hairpin Polyamide Platinum Complexes
title_full Synthesis of DNA-Sequence-Selective Hairpin Polyamide Platinum Complexes
title_fullStr Synthesis of DNA-Sequence-Selective Hairpin Polyamide Platinum Complexes
title_full_unstemmed Synthesis of DNA-Sequence-Selective Hairpin Polyamide Platinum Complexes
title_short Synthesis of DNA-Sequence-Selective Hairpin Polyamide Platinum Complexes
title_sort Synthesis of DNA-Sequence-Selective Hairpin Polyamide Platinum Complexes
url http://hdl.handle.net/10725/3496
http://dx.doi.org/10.1002/chem.200601486
http://onlinelibrary.wiley.com/doi/10.1002/chem.200601486/full