Fluorescence of 6-methoxyquinoline, quinine, and quinidine in aqueous media

The absorption and fluorescence spectra of 6-methoxy-quinoline, quinine, and quinidine were studied as a continuous function of pH. 6-Methoxyquinoline is a stronger base in the lowest excited singlet state, as reflected by the pH dependence of its fluorescence. The latter is used to calculate the ra...

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Main Author: Capomacchia, Anthony C. (author)
Other Authors: Threatte, Rose Marie (author), Schulman, Stephen C. (author)
Format: article
Published: 1974
Online Access:http://hdl.handle.net/10725/6333
http://dx.doi.org/10.1002/jps.2600630615
http://libraries.lau.edu.lb/research/laur/terms-of-use/articles.php
http://onlinelibrary.wiley.com/doi/10.1002/jps.2600630615/full
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author Capomacchia, Anthony C.
author2 Threatte, Rose Marie
Schulman, Stephen C.
author2_role author
author
author_facet Capomacchia, Anthony C.
Threatte, Rose Marie
Schulman, Stephen C.
author_role author
dc.creator.none.fl_str_mv Capomacchia, Anthony C.
Threatte, Rose Marie
Schulman, Stephen C.
dc.date.none.fl_str_mv 1974
2017-10-17T11:36:27Z
2017-10-17T11:36:27Z
2017-10-17
dc.identifier.none.fl_str_mv 1520-6017
http://hdl.handle.net/10725/6333
http://dx.doi.org/10.1002/jps.2600630615
Schulman, S. G., Threatte, R. M., Capomacchia, A. C., & Paul, W. L. (1974). Fluorescence of 6‐methoxyquinoline, quinine, and quinidine in aqueous media. Journal of pharmaceutical sciences, 63(6), 876-880.
http://libraries.lau.edu.lb/research/laur/terms-of-use/articles.php
http://onlinelibrary.wiley.com/doi/10.1002/jps.2600630615/full
dc.language.none.fl_str_mv en
dc.relation.none.fl_str_mv Journal of Pharmaceutical Sciences
dc.rights.*.fl_str_mv info:eu-repo/semantics/openAccess
dc.title.none.fl_str_mv Fluorescence of 6-methoxyquinoline, quinine, and quinidine in aqueous media
dc.type.none.fl_str_mv Article
info:eu-repo/semantics/publishedVersion
info:eu-repo/semantics/article
description The absorption and fluorescence spectra of 6-methoxy-quinoline, quinine, and quinidine were studied as a continuous function of pH. 6-Methoxyquinoline is a stronger base in the lowest excited singlet state, as reflected by the pH dependence of its fluorescence. The latter is used to calculate the rates and equilibria of proton exchange in the excited state. Quinine and quinidine, however, do not protonate during the lifetimes of their excited states, an observation attributed to the lower basicity of their aromatic heterocyclic nitrogen than that in 6-methoxyquinoline. The differences in basic properties between the alkaloids and 6-methoxyquinoline are employed to infer the ketonic character of the quinolinemethanol group of the alkaloids and the existence of an intramolecular hydrogen bond in quinine but not in quinidine.
eu_rights_str_mv openAccess
format article
id LAURepo_c83fbbfbd081e2be6ff07644706fd0b5
identifier_str_mv 1520-6017
Schulman, S. G., Threatte, R. M., Capomacchia, A. C., & Paul, W. L. (1974). Fluorescence of 6‐methoxyquinoline, quinine, and quinidine in aqueous media. Journal of pharmaceutical sciences, 63(6), 876-880.
language_invalid_str_mv en
network_acronym_str LAURepo
network_name_str Lebanese American University repository
oai_identifier_str oai:laur.lau.edu.lb:10725/6333
publishDate 1974
repository.mail.fl_str_mv
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spelling Fluorescence of 6-methoxyquinoline, quinine, and quinidine in aqueous mediaCapomacchia, Anthony C.Threatte, Rose MarieSchulman, Stephen C.The absorption and fluorescence spectra of 6-methoxy-quinoline, quinine, and quinidine were studied as a continuous function of pH. 6-Methoxyquinoline is a stronger base in the lowest excited singlet state, as reflected by the pH dependence of its fluorescence. The latter is used to calculate the rates and equilibria of proton exchange in the excited state. Quinine and quinidine, however, do not protonate during the lifetimes of their excited states, an observation attributed to the lower basicity of their aromatic heterocyclic nitrogen than that in 6-methoxyquinoline. The differences in basic properties between the alkaloids and 6-methoxyquinoline are employed to infer the ketonic character of the quinolinemethanol group of the alkaloids and the existence of an intramolecular hydrogen bond in quinine but not in quinidine.PublishedN/A2017-10-17T11:36:27Z2017-10-17T11:36:27Z19742017-10-17Articleinfo:eu-repo/semantics/publishedVersioninfo:eu-repo/semantics/article1520-6017http://hdl.handle.net/10725/6333http://dx.doi.org/10.1002/jps.2600630615Schulman, S. G., Threatte, R. M., Capomacchia, A. C., & Paul, W. L. (1974). Fluorescence of 6‐methoxyquinoline, quinine, and quinidine in aqueous media. Journal of pharmaceutical sciences, 63(6), 876-880.http://libraries.lau.edu.lb/research/laur/terms-of-use/articles.phphttp://onlinelibrary.wiley.com/doi/10.1002/jps.2600630615/fullenJournal of Pharmaceutical Sciencesinfo:eu-repo/semantics/openAccessoai:laur.lau.edu.lb:10725/63332021-03-19T10:03:25Z
spellingShingle Fluorescence of 6-methoxyquinoline, quinine, and quinidine in aqueous media
Capomacchia, Anthony C.
status_str publishedVersion
title Fluorescence of 6-methoxyquinoline, quinine, and quinidine in aqueous media
title_full Fluorescence of 6-methoxyquinoline, quinine, and quinidine in aqueous media
title_fullStr Fluorescence of 6-methoxyquinoline, quinine, and quinidine in aqueous media
title_full_unstemmed Fluorescence of 6-methoxyquinoline, quinine, and quinidine in aqueous media
title_short Fluorescence of 6-methoxyquinoline, quinine, and quinidine in aqueous media
title_sort Fluorescence of 6-methoxyquinoline, quinine, and quinidine in aqueous media
url http://hdl.handle.net/10725/6333
http://dx.doi.org/10.1002/jps.2600630615
http://libraries.lau.edu.lb/research/laur/terms-of-use/articles.php
http://onlinelibrary.wiley.com/doi/10.1002/jps.2600630615/full