Strategies for the production of long-acting therapeutics and efficient drug delivery for cancer treatment

<p>Protein therapeutics play a significant role in treating many diseases. They, however, suffer from patient’s proteases degradation and antibody neutralization which lead to short plasma half-lives. One of the ways to overcome these pitfalls is the frequent injection of the drug albeit at th...

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Main Author: Alanod D. AlQahtani (18805930) (author)
Other Authors: David O’Connor (108088) (author), Alexander Domling (18805927) (author), Sayed K. Goda (5146160) (author)
Published: 2019
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author Alanod D. AlQahtani (18805930)
author2 David O’Connor (108088)
Alexander Domling (18805927)
Sayed K. Goda (5146160)
author2_role author
author
author
author_facet Alanod D. AlQahtani (18805930)
David O’Connor (108088)
Alexander Domling (18805927)
Sayed K. Goda (5146160)
author_role author
dc.creator.none.fl_str_mv Alanod D. AlQahtani (18805930)
David O’Connor (108088)
Alexander Domling (18805927)
Sayed K. Goda (5146160)
dc.date.none.fl_str_mv 2019-05-01T00:00:00Z
dc.identifier.none.fl_str_mv 10.1016/j.biopha.2019.108750
dc.relation.none.fl_str_mv https://figshare.com/articles/journal_contribution/Strategies_for_the_production_of_long-acting_therapeutics_and_efficient_drug_delivery_for_cancer_treatment/26015830
dc.rights.none.fl_str_mv CC BY 4.0
info:eu-repo/semantics/openAccess
dc.subject.none.fl_str_mv Biomedical and clinical sciences
Medical biotechnology
Ophthalmology and optometry
Pharmacology and pharmaceutical sciences
PEGylations
Human serum albumin
Targeted cancer cells
Drug delivery
Half-life extension
Protein immunogenicity
dc.title.none.fl_str_mv Strategies for the production of long-acting therapeutics and efficient drug delivery for cancer treatment
dc.type.none.fl_str_mv Text
Journal contribution
info:eu-repo/semantics/publishedVersion
text
contribution to journal
description <p>Protein therapeutics play a significant role in treating many diseases. They, however, suffer from patient’s proteases degradation and antibody neutralization which lead to short plasma half-lives. One of the ways to overcome these pitfalls is the frequent injection of the drug albeit at the cost of patient compliance which affects the quality of life of patients. There are several techniques available to extend the half-life of therapeutics. Two of the most common protocols are PEGylation and fusion with human serum albumin. These two techniques improve stability, reduce immunogenicity, and increase drug resistance to proteases. These factors lead to the reduction of injection frequency which increases patient compliance and improve quality of life. Both techniques have already been used in many FDA approved drugs. This review describes many technologies to produce long-acting drugs with the attention of PEGylation and the genetic fusion with human serum albumin. The report also discusses the latest modified therapeutics in the field and their application in cancer therapy. We compare the modification methods and discuss the pitfalls of these modified drugs.</p><h2>Other Information</h2> <p> Published in: Biomedicine & Pharmacotherapy<br> License: <a href="http://creativecommons.org/licenses/by/4.0/" target="_blank">http://creativecommons.org/licenses/by/4.0/</a><br>See article on publisher's website: <a href="https://dx.doi.org/10.1016/j.biopha.2019.108750" target="_blank">https://dx.doi.org/10.1016/j.biopha.2019.108750</a></p>
eu_rights_str_mv openAccess
id Manara2_212fd7846ce35d8e0a53b79e847e52e8
identifier_str_mv 10.1016/j.biopha.2019.108750
network_acronym_str Manara2
network_name_str Manara2
oai_identifier_str oai:figshare.com:article/26015830
publishDate 2019
repository.mail.fl_str_mv
repository.name.fl_str_mv
repository_id_str
rights_invalid_str_mv CC BY 4.0
spelling Strategies for the production of long-acting therapeutics and efficient drug delivery for cancer treatmentAlanod D. AlQahtani (18805930)David O’Connor (108088)Alexander Domling (18805927)Sayed K. Goda (5146160)Biomedical and clinical sciencesMedical biotechnologyOphthalmology and optometryPharmacology and pharmaceutical sciencesPEGylationsHuman serum albuminTargeted cancer cellsDrug deliveryHalf-life extensionProtein immunogenicity<p>Protein therapeutics play a significant role in treating many diseases. They, however, suffer from patient’s proteases degradation and antibody neutralization which lead to short plasma half-lives. One of the ways to overcome these pitfalls is the frequent injection of the drug albeit at the cost of patient compliance which affects the quality of life of patients. There are several techniques available to extend the half-life of therapeutics. Two of the most common protocols are PEGylation and fusion with human serum albumin. These two techniques improve stability, reduce immunogenicity, and increase drug resistance to proteases. These factors lead to the reduction of injection frequency which increases patient compliance and improve quality of life. Both techniques have already been used in many FDA approved drugs. This review describes many technologies to produce long-acting drugs with the attention of PEGylation and the genetic fusion with human serum albumin. The report also discusses the latest modified therapeutics in the field and their application in cancer therapy. We compare the modification methods and discuss the pitfalls of these modified drugs.</p><h2>Other Information</h2> <p> Published in: Biomedicine & Pharmacotherapy<br> License: <a href="http://creativecommons.org/licenses/by/4.0/" target="_blank">http://creativecommons.org/licenses/by/4.0/</a><br>See article on publisher's website: <a href="https://dx.doi.org/10.1016/j.biopha.2019.108750" target="_blank">https://dx.doi.org/10.1016/j.biopha.2019.108750</a></p>2019-05-01T00:00:00ZTextJournal contributioninfo:eu-repo/semantics/publishedVersiontextcontribution to journal10.1016/j.biopha.2019.108750https://figshare.com/articles/journal_contribution/Strategies_for_the_production_of_long-acting_therapeutics_and_efficient_drug_delivery_for_cancer_treatment/26015830CC BY 4.0info:eu-repo/semantics/openAccessoai:figshare.com:article/260158302019-05-01T00:00:00Z
spellingShingle Strategies for the production of long-acting therapeutics and efficient drug delivery for cancer treatment
Alanod D. AlQahtani (18805930)
Biomedical and clinical sciences
Medical biotechnology
Ophthalmology and optometry
Pharmacology and pharmaceutical sciences
PEGylations
Human serum albumin
Targeted cancer cells
Drug delivery
Half-life extension
Protein immunogenicity
status_str publishedVersion
title Strategies for the production of long-acting therapeutics and efficient drug delivery for cancer treatment
title_full Strategies for the production of long-acting therapeutics and efficient drug delivery for cancer treatment
title_fullStr Strategies for the production of long-acting therapeutics and efficient drug delivery for cancer treatment
title_full_unstemmed Strategies for the production of long-acting therapeutics and efficient drug delivery for cancer treatment
title_short Strategies for the production of long-acting therapeutics and efficient drug delivery for cancer treatment
title_sort Strategies for the production of long-acting therapeutics and efficient drug delivery for cancer treatment
topic Biomedical and clinical sciences
Medical biotechnology
Ophthalmology and optometry
Pharmacology and pharmaceutical sciences
PEGylations
Human serum albumin
Targeted cancer cells
Drug delivery
Half-life extension
Protein immunogenicity