Probing the effect of clustering on EphA2 receptor signaling efficiency by subcellular control of ligand-receptor mobility

<div><p>Clustering of ligand:receptor complexes on the cell membrane is widely presumed to have functional consequences for subsequent signal transduction. However, it is experimentally challenging to selectively manipulate receptor clustering without altering other biochemical aspects o...

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محفوظ في:
التفاصيل البيبلوغرافية
المؤلف الرئيسي: Zhongwen Chen (770401) (author)
مؤلفون آخرون: Dongmyung Oh (2361895) (author), Kabir Hassan Biswas (18595561) (author), Ronen Zaidel-Bar (711501) (author), Jay T Groves (18595564) (author)
منشور في: 2021
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author Zhongwen Chen (770401)
author2 Dongmyung Oh (2361895)
Kabir Hassan Biswas (18595561)
Ronen Zaidel-Bar (711501)
Jay T Groves (18595564)
author2_role author
author
author
author
author_facet Zhongwen Chen (770401)
Dongmyung Oh (2361895)
Kabir Hassan Biswas (18595561)
Ronen Zaidel-Bar (711501)
Jay T Groves (18595564)
author_role author
dc.creator.none.fl_str_mv Zhongwen Chen (770401)
Dongmyung Oh (2361895)
Kabir Hassan Biswas (18595561)
Ronen Zaidel-Bar (711501)
Jay T Groves (18595564)
dc.date.none.fl_str_mv 2021-08-20T03:00:00Z
dc.identifier.none.fl_str_mv 10.7554/elife.67379
dc.relation.none.fl_str_mv https://figshare.com/articles/journal_contribution/Probing_the_effect_of_clustering_on_EphA2_receptor_signaling_efficiency_by_subcellular_control_of_ligand-receptor_mobility/25877974
dc.rights.none.fl_str_mv CC BY 4.0
info:eu-repo/semantics/openAccess
dc.subject.none.fl_str_mv Biological sciences
Biochemistry and cell biology
Ligand-receptor complexes
Cell membrane
Signal transduction
Receptor clustering
Microfabrication
Substrates
Mobile ligands
dc.title.none.fl_str_mv Probing the effect of clustering on EphA2 receptor signaling efficiency by subcellular control of ligand-receptor mobility
dc.type.none.fl_str_mv Text
Journal contribution
info:eu-repo/semantics/publishedVersion
text
contribution to journal
description <div><p>Clustering of ligand:receptor complexes on the cell membrane is widely presumed to have functional consequences for subsequent signal transduction. However, it is experimentally challenging to selectively manipulate receptor clustering without altering other biochemical aspects of the cellular system. Here, we develop a microfabrication strategy to produce substrates displaying mobile and immobile ligands that are separated by roughly 1 µm, and thus experience an identical cytoplasmic signaling state, enabling precision comparison of downstream signaling reactions. Applying this approach to characterize the ephrinA1:EphA2 signaling system reveals that EphA2 clustering enhances both receptor phosphorylation and downstream signaling activity. Single-molecule imaging clearly resolves increased molecular binding dwell times at EphA2 clusters for both Grb2:SOS and NCK:N-WASP signaling modules. This type of intracellular comparison enables a substantially higher degree of quantitative analysis than is possible when comparisons must be made between different cells and essentially eliminates the effects of cellular response to ligand manipulation.</p><p> </p></div><h2>Other Information</h2> <p> Published in: eLife<br> License: <a href="http://creativecommons.org/licenses/by/4.0/" target="_blank">http://creativecommons.org/licenses/by/4.0/</a><br>See article on publisher's website: <a href="https://dx.doi.org/10.7554/elife.67379" target="_blank">https://dx.doi.org/10.7554/elife.67379</a></p>
eu_rights_str_mv openAccess
id Manara2_242b7534abf02e753a219f488b124ad0
identifier_str_mv 10.7554/elife.67379
network_acronym_str Manara2
network_name_str Manara2
oai_identifier_str oai:figshare.com:article/25877974
publishDate 2021
repository.mail.fl_str_mv
repository.name.fl_str_mv
repository_id_str
rights_invalid_str_mv CC BY 4.0
spelling Probing the effect of clustering on EphA2 receptor signaling efficiency by subcellular control of ligand-receptor mobilityZhongwen Chen (770401)Dongmyung Oh (2361895)Kabir Hassan Biswas (18595561)Ronen Zaidel-Bar (711501)Jay T Groves (18595564)Biological sciencesBiochemistry and cell biologyLigand-receptor complexesCell membraneSignal transductionReceptor clusteringMicrofabricationSubstratesMobile ligands<div><p>Clustering of ligand:receptor complexes on the cell membrane is widely presumed to have functional consequences for subsequent signal transduction. However, it is experimentally challenging to selectively manipulate receptor clustering without altering other biochemical aspects of the cellular system. Here, we develop a microfabrication strategy to produce substrates displaying mobile and immobile ligands that are separated by roughly 1 µm, and thus experience an identical cytoplasmic signaling state, enabling precision comparison of downstream signaling reactions. Applying this approach to characterize the ephrinA1:EphA2 signaling system reveals that EphA2 clustering enhances both receptor phosphorylation and downstream signaling activity. Single-molecule imaging clearly resolves increased molecular binding dwell times at EphA2 clusters for both Grb2:SOS and NCK:N-WASP signaling modules. This type of intracellular comparison enables a substantially higher degree of quantitative analysis than is possible when comparisons must be made between different cells and essentially eliminates the effects of cellular response to ligand manipulation.</p><p> </p></div><h2>Other Information</h2> <p> Published in: eLife<br> License: <a href="http://creativecommons.org/licenses/by/4.0/" target="_blank">http://creativecommons.org/licenses/by/4.0/</a><br>See article on publisher's website: <a href="https://dx.doi.org/10.7554/elife.67379" target="_blank">https://dx.doi.org/10.7554/elife.67379</a></p>2021-08-20T03:00:00ZTextJournal contributioninfo:eu-repo/semantics/publishedVersiontextcontribution to journal10.7554/elife.67379https://figshare.com/articles/journal_contribution/Probing_the_effect_of_clustering_on_EphA2_receptor_signaling_efficiency_by_subcellular_control_of_ligand-receptor_mobility/25877974CC BY 4.0info:eu-repo/semantics/openAccessoai:figshare.com:article/258779742021-08-20T03:00:00Z
spellingShingle Probing the effect of clustering on EphA2 receptor signaling efficiency by subcellular control of ligand-receptor mobility
Zhongwen Chen (770401)
Biological sciences
Biochemistry and cell biology
Ligand-receptor complexes
Cell membrane
Signal transduction
Receptor clustering
Microfabrication
Substrates
Mobile ligands
status_str publishedVersion
title Probing the effect of clustering on EphA2 receptor signaling efficiency by subcellular control of ligand-receptor mobility
title_full Probing the effect of clustering on EphA2 receptor signaling efficiency by subcellular control of ligand-receptor mobility
title_fullStr Probing the effect of clustering on EphA2 receptor signaling efficiency by subcellular control of ligand-receptor mobility
title_full_unstemmed Probing the effect of clustering on EphA2 receptor signaling efficiency by subcellular control of ligand-receptor mobility
title_short Probing the effect of clustering on EphA2 receptor signaling efficiency by subcellular control of ligand-receptor mobility
title_sort Probing the effect of clustering on EphA2 receptor signaling efficiency by subcellular control of ligand-receptor mobility
topic Biological sciences
Biochemistry and cell biology
Ligand-receptor complexes
Cell membrane
Signal transduction
Receptor clustering
Microfabrication
Substrates
Mobile ligands