In vitro Anti-Helicobacter pylori Activity of Capsaicin

<p dir="ltr">Worldwide, peptic ulcer and gastritis considered to be one of the biggest health challenge, <i>Helicobacter pylori</i> is responsible for more than eighty percent of chronic active gastritis where continual infection remains for decennary. However, the succes...

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المؤلف الرئيسي: Department of Pharmaceutical Sciences, Faculty of Pharmacy, University of Jordan, Amman, Jordan. (19672696) (author)
مؤلفون آخرون: Isra Tayseer (19672699) (author), Talal Aburjai (19672702) (author), Luay Abu-Qatouseh (12106047) (author), Faculty of Pharmacy, Department of Biomedical Sciences, University of Petra, Amman, Jordan. (19672708) (author), Nehaya AL-Karabieh (19672711) (author), Department of Plant Protection, School of Agriculture, The University of Jordan, Amman, Jordan. (19672714) (author), Wesam Ahmed (4870942) (author), Ali Al-Samydai (18176017) (author)
منشور في: 2020
الموضوعات:
الوسوم: إضافة وسم
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author Department of Pharmaceutical Sciences, Faculty of Pharmacy, University of Jordan, Amman, Jordan. (19672696)
author2 Isra Tayseer (19672699)
Talal Aburjai (19672702)
Luay Abu-Qatouseh (12106047)
Faculty of Pharmacy, Department of Biomedical Sciences, University of Petra, Amman, Jordan. (19672708)
Nehaya AL-Karabieh (19672711)
Department of Plant Protection, School of Agriculture, The University of Jordan, Amman, Jordan. (19672714)
Wesam Ahmed (4870942)
Ali Al-Samydai (18176017)
author2_role author
author
author
author
author
author
author
author
author_facet Department of Pharmaceutical Sciences, Faculty of Pharmacy, University of Jordan, Amman, Jordan. (19672696)
Isra Tayseer (19672699)
Talal Aburjai (19672702)
Luay Abu-Qatouseh (12106047)
Faculty of Pharmacy, Department of Biomedical Sciences, University of Petra, Amman, Jordan. (19672708)
Nehaya AL-Karabieh (19672711)
Department of Plant Protection, School of Agriculture, The University of Jordan, Amman, Jordan. (19672714)
Wesam Ahmed (4870942)
Ali Al-Samydai (18176017)
author_role author
dc.creator.none.fl_str_mv Department of Pharmaceutical Sciences, Faculty of Pharmacy, University of Jordan, Amman, Jordan. (19672696)
Isra Tayseer (19672699)
Talal Aburjai (19672702)
Luay Abu-Qatouseh (12106047)
Faculty of Pharmacy, Department of Biomedical Sciences, University of Petra, Amman, Jordan. (19672708)
Nehaya AL-Karabieh (19672711)
Department of Plant Protection, School of Agriculture, The University of Jordan, Amman, Jordan. (19672714)
Wesam Ahmed (4870942)
Ali Al-Samydai (18176017)
dc.date.none.fl_str_mv 2020-03-21T06:00:00Z
dc.identifier.none.fl_str_mv 10.22207/jpam.14.1.29
dc.relation.none.fl_str_mv https://figshare.com/articles/journal_contribution/In_vitro_Anti-Helicobacter_pylori_Activity_of_Capsaicin/27021688
dc.rights.none.fl_str_mv CC BY 4.0
info:eu-repo/semantics/openAccess
dc.subject.none.fl_str_mv Biological sciences
Microbiology
Biomedical and clinical sciences
Pharmacology and pharmaceutical sciences
H. pylori
Capsaicin
Spices
Synergism
dc.title.none.fl_str_mv In vitro Anti-Helicobacter pylori Activity of Capsaicin
dc.type.none.fl_str_mv Text
Journal contribution
info:eu-repo/semantics/publishedVersion
text
contribution to journal
description <p dir="ltr">Worldwide, peptic ulcer and gastritis considered to be one of the biggest health challenge, <i>Helicobacter pylori</i> is responsible for more than eighty percent of chronic active gastritis where continual infection remains for decennary. However, the success of commercially available drugs for the management of <i>H. pylori</i> has overwhelmed by antibiotic-resistant strains, especially, metronidazole and clarithromycin, therefore, an urgent need arise to search for new options for treatment with enhanced anti- <i>H. pylori</i> activities, while being less toxic to human cells. Naturally occurring plant products, including spices, are one of these strategies that showed activity against <i>H. pylori</i>. Present study aim to test the antibacterial activity of capsaicin and other pure plant-derived compounds against a standard (NCTC 11916) H. pylori strain In vitro and to test for possible synergistic effect when combined with conventional therapy. Capsaicin shows good antibacterial activity on regular antimicrobial sensitivity testing methods (Anti-MSTM) and titration checkerboard assay MIC (0.0625 mg/ml), whereas piperine MIC was (0.125 mg/ml). While for curcumin no inhibition was found. The strain was found to be resistant to metronidazole with (MIC=250 μg/ml). When combining capsaicin with metronidazole, (FIC) Fractional inhibitory concentration values shown a synergistic effect, While the additive effect was found for capsaicin combination with piperine. Our obtained data indicate that capsaicin possesses promising anti <i>H. pylori</i> bioactivity and synergistic activity when combined with metronidazole but more work is necessary to examine the mechanisms by which these happened. Furthermore, it is necessary to ensure its activity against <i>H. pylori</i> <i>In vivo</i> and clinical settings.</p><h2>Other Information</h2><p dir="ltr">Published in: Journal of Pure and Applied Microbiology<br>License: <a href="https://creativecommons.org/licenses/by/4.0/" target="_blank">https://creativecommons.org/licenses/by/4.0/</a><br>See article on publisher's website: <a href="https://dx.doi.org/10.22207/jpam.14.1.29" target="_blank">https://dx.doi.org/10.22207/jpam.14.1.29</a></p>
eu_rights_str_mv openAccess
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network_acronym_str Manara2
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spelling In vitro Anti-Helicobacter pylori Activity of CapsaicinDepartment of Pharmaceutical Sciences, Faculty of Pharmacy, University of Jordan, Amman, Jordan. (19672696)Isra Tayseer (19672699)Talal Aburjai (19672702)Luay Abu-Qatouseh (12106047)Faculty of Pharmacy, Department of Biomedical Sciences, University of Petra, Amman, Jordan. (19672708)Nehaya AL-Karabieh (19672711)Department of Plant Protection, School of Agriculture, The University of Jordan, Amman, Jordan. (19672714)Wesam Ahmed (4870942)Ali Al-Samydai (18176017)Biological sciencesMicrobiologyBiomedical and clinical sciencesPharmacology and pharmaceutical sciencesH. pyloriCapsaicinSpicesSynergism<p dir="ltr">Worldwide, peptic ulcer and gastritis considered to be one of the biggest health challenge, <i>Helicobacter pylori</i> is responsible for more than eighty percent of chronic active gastritis where continual infection remains for decennary. However, the success of commercially available drugs for the management of <i>H. pylori</i> has overwhelmed by antibiotic-resistant strains, especially, metronidazole and clarithromycin, therefore, an urgent need arise to search for new options for treatment with enhanced anti- <i>H. pylori</i> activities, while being less toxic to human cells. Naturally occurring plant products, including spices, are one of these strategies that showed activity against <i>H. pylori</i>. Present study aim to test the antibacterial activity of capsaicin and other pure plant-derived compounds against a standard (NCTC 11916) H. pylori strain In vitro and to test for possible synergistic effect when combined with conventional therapy. Capsaicin shows good antibacterial activity on regular antimicrobial sensitivity testing methods (Anti-MSTM) and titration checkerboard assay MIC (0.0625 mg/ml), whereas piperine MIC was (0.125 mg/ml). While for curcumin no inhibition was found. The strain was found to be resistant to metronidazole with (MIC=250 μg/ml). When combining capsaicin with metronidazole, (FIC) Fractional inhibitory concentration values shown a synergistic effect, While the additive effect was found for capsaicin combination with piperine. Our obtained data indicate that capsaicin possesses promising anti <i>H. pylori</i> bioactivity and synergistic activity when combined with metronidazole but more work is necessary to examine the mechanisms by which these happened. Furthermore, it is necessary to ensure its activity against <i>H. pylori</i> <i>In vivo</i> and clinical settings.</p><h2>Other Information</h2><p dir="ltr">Published in: Journal of Pure and Applied Microbiology<br>License: <a href="https://creativecommons.org/licenses/by/4.0/" target="_blank">https://creativecommons.org/licenses/by/4.0/</a><br>See article on publisher's website: <a href="https://dx.doi.org/10.22207/jpam.14.1.29" target="_blank">https://dx.doi.org/10.22207/jpam.14.1.29</a></p>2020-03-21T06:00:00ZTextJournal contributioninfo:eu-repo/semantics/publishedVersiontextcontribution to journal10.22207/jpam.14.1.29https://figshare.com/articles/journal_contribution/In_vitro_Anti-Helicobacter_pylori_Activity_of_Capsaicin/27021688CC BY 4.0info:eu-repo/semantics/openAccessoai:figshare.com:article/270216882020-03-21T06:00:00Z
spellingShingle In vitro Anti-Helicobacter pylori Activity of Capsaicin
Department of Pharmaceutical Sciences, Faculty of Pharmacy, University of Jordan, Amman, Jordan. (19672696)
Biological sciences
Microbiology
Biomedical and clinical sciences
Pharmacology and pharmaceutical sciences
H. pylori
Capsaicin
Spices
Synergism
status_str publishedVersion
title In vitro Anti-Helicobacter pylori Activity of Capsaicin
title_full In vitro Anti-Helicobacter pylori Activity of Capsaicin
title_fullStr In vitro Anti-Helicobacter pylori Activity of Capsaicin
title_full_unstemmed In vitro Anti-Helicobacter pylori Activity of Capsaicin
title_short In vitro Anti-Helicobacter pylori Activity of Capsaicin
title_sort In vitro Anti-Helicobacter pylori Activity of Capsaicin
topic Biological sciences
Microbiology
Biomedical and clinical sciences
Pharmacology and pharmaceutical sciences
H. pylori
Capsaicin
Spices
Synergism