Use of Animal Models for Investigating Cardioprotective Roles of SGLT2 Inhibitors

<p dir="ltr">Sodium-glucose co-transporter 2 (SGLT2) inhibitors represent one type of new-generation type 2 diabetes (T2DM) drug treatment. The mechanism of action of an SGLT2 inhibitor (SGLT2i) in treating T2DM depends on lowering blood glucose levels effectively via increasing the...

Full description

Saved in:
Bibliographic Details
Main Author: Najlaa A. Al Thani (17788493) (author)
Other Authors: Maram Hasan (6672440) (author), Huseyin C. Yalcin (6695099) (author)
Published: 2023
Subjects:
Tags: Add Tag
No Tags, Be the first to tag this record!
_version_ 1864513530543210496
author Najlaa A. Al Thani (17788493)
author2 Maram Hasan (6672440)
Huseyin C. Yalcin (6695099)
author2_role author
author
author_facet Najlaa A. Al Thani (17788493)
Maram Hasan (6672440)
Huseyin C. Yalcin (6695099)
author_role author
dc.creator.none.fl_str_mv Najlaa A. Al Thani (17788493)
Maram Hasan (6672440)
Huseyin C. Yalcin (6695099)
dc.date.none.fl_str_mv 2023-04-13T03:00:00Z
dc.identifier.none.fl_str_mv 10.1007/s12265-023-10379-5
dc.relation.none.fl_str_mv https://figshare.com/articles/journal_contribution/Use_of_Animal_Models_for_Investigating_Cardioprotective_Roles_of_SGLT2_Inhibitors/24998591
dc.rights.none.fl_str_mv CC BY 4.0
info:eu-repo/semantics/openAccess
dc.subject.none.fl_str_mv Biomedical and clinical sciences
Cardiovascular medicine and haematology
Clinical sciences
Pharmacology and pharmaceutical sciences
SLGT2
Diabetes
Heart failure
Cardioprotection
Glifozins
Empaglifozin
Canaglifozin
Animal models
dc.title.none.fl_str_mv Use of Animal Models for Investigating Cardioprotective Roles of SGLT2 Inhibitors
dc.type.none.fl_str_mv Text
Journal contribution
info:eu-repo/semantics/publishedVersion
text
contribution to journal
description <p dir="ltr">Sodium-glucose co-transporter 2 (SGLT2) inhibitors represent one type of new-generation type 2 diabetes (T2DM) drug treatment. The mechanism of action of an SGLT2 inhibitor (SGLT2i) in treating T2DM depends on lowering blood glucose levels effectively via increasing the glomerular excretion of glucose. A good number of randomized clinical trials revealed that SGLT2is significantly prevented heart failure (HF) and cardiovascular death in T2DM patients. Despite ongoing clinical trials in HF patients without T2DM, there have been a limited number of translational studies on the cardioprotective properties of SGLT2is. As the cellular mechanism behind the cardiac benefits of SGLT2is is still to be elucidated, animal models are used to better understand the pathways behind the cardioprotective mechanism of SGLT2i. In this review, we summarize the animal models constructed to study the cardioprotective mechanisms of SGLT2is to help deliver a more comprehensive understanding of the in vivo work that has been done in this field and to help select the most optimal animal model to use when studying the different cardioprotective effects of SGLT2is.</p><h2>Other Information</h2><p dir="ltr">Published in: Journal of Cardiovascular Translational Research<br>License: <a href="https://creativecommons.org/licenses/by/4.0" target="_blank">https://creativecommons.org/licenses/by/4.0</a><br>See article on publisher's website: <a href="https://dx.doi.org/10.1007/s12265-023-10379-5" target="_blank">https://dx.doi.org/10.1007/s12265-023-10379-5</a></p>
eu_rights_str_mv openAccess
id Manara2_7373cde6e273753401fccc0611a08d03
identifier_str_mv 10.1007/s12265-023-10379-5
network_acronym_str Manara2
network_name_str Manara2
oai_identifier_str oai:figshare.com:article/24998591
publishDate 2023
repository.mail.fl_str_mv
repository.name.fl_str_mv
repository_id_str
rights_invalid_str_mv CC BY 4.0
spelling Use of Animal Models for Investigating Cardioprotective Roles of SGLT2 InhibitorsNajlaa A. Al Thani (17788493)Maram Hasan (6672440)Huseyin C. Yalcin (6695099)Biomedical and clinical sciencesCardiovascular medicine and haematologyClinical sciencesPharmacology and pharmaceutical sciencesSLGT2DiabetesHeart failureCardioprotectionGlifozinsEmpaglifozinCanaglifozinAnimal models<p dir="ltr">Sodium-glucose co-transporter 2 (SGLT2) inhibitors represent one type of new-generation type 2 diabetes (T2DM) drug treatment. The mechanism of action of an SGLT2 inhibitor (SGLT2i) in treating T2DM depends on lowering blood glucose levels effectively via increasing the glomerular excretion of glucose. A good number of randomized clinical trials revealed that SGLT2is significantly prevented heart failure (HF) and cardiovascular death in T2DM patients. Despite ongoing clinical trials in HF patients without T2DM, there have been a limited number of translational studies on the cardioprotective properties of SGLT2is. As the cellular mechanism behind the cardiac benefits of SGLT2is is still to be elucidated, animal models are used to better understand the pathways behind the cardioprotective mechanism of SGLT2i. In this review, we summarize the animal models constructed to study the cardioprotective mechanisms of SGLT2is to help deliver a more comprehensive understanding of the in vivo work that has been done in this field and to help select the most optimal animal model to use when studying the different cardioprotective effects of SGLT2is.</p><h2>Other Information</h2><p dir="ltr">Published in: Journal of Cardiovascular Translational Research<br>License: <a href="https://creativecommons.org/licenses/by/4.0" target="_blank">https://creativecommons.org/licenses/by/4.0</a><br>See article on publisher's website: <a href="https://dx.doi.org/10.1007/s12265-023-10379-5" target="_blank">https://dx.doi.org/10.1007/s12265-023-10379-5</a></p>2023-04-13T03:00:00ZTextJournal contributioninfo:eu-repo/semantics/publishedVersiontextcontribution to journal10.1007/s12265-023-10379-5https://figshare.com/articles/journal_contribution/Use_of_Animal_Models_for_Investigating_Cardioprotective_Roles_of_SGLT2_Inhibitors/24998591CC BY 4.0info:eu-repo/semantics/openAccessoai:figshare.com:article/249985912023-04-13T03:00:00Z
spellingShingle Use of Animal Models for Investigating Cardioprotective Roles of SGLT2 Inhibitors
Najlaa A. Al Thani (17788493)
Biomedical and clinical sciences
Cardiovascular medicine and haematology
Clinical sciences
Pharmacology and pharmaceutical sciences
SLGT2
Diabetes
Heart failure
Cardioprotection
Glifozins
Empaglifozin
Canaglifozin
Animal models
status_str publishedVersion
title Use of Animal Models for Investigating Cardioprotective Roles of SGLT2 Inhibitors
title_full Use of Animal Models for Investigating Cardioprotective Roles of SGLT2 Inhibitors
title_fullStr Use of Animal Models for Investigating Cardioprotective Roles of SGLT2 Inhibitors
title_full_unstemmed Use of Animal Models for Investigating Cardioprotective Roles of SGLT2 Inhibitors
title_short Use of Animal Models for Investigating Cardioprotective Roles of SGLT2 Inhibitors
title_sort Use of Animal Models for Investigating Cardioprotective Roles of SGLT2 Inhibitors
topic Biomedical and clinical sciences
Cardiovascular medicine and haematology
Clinical sciences
Pharmacology and pharmaceutical sciences
SLGT2
Diabetes
Heart failure
Cardioprotection
Glifozins
Empaglifozin
Canaglifozin
Animal models