Curcumin and Derivatives in Nanoformulations with Therapeutic Potential on Colorectal Cancer

<p>There is growing concern in the rise of colorectal cancer (CRC) cases globally, and with this rise is the presentation of drug resistance. Like other cancers, current treatment options are either invasive or manifest severe side effects. Thus, there is a move towards implementing safer trea...

وصف كامل

محفوظ في:
التفاصيل البيبلوغرافية
المؤلف الرئيسي: Sourour Idoudi (14153457) (author)
مؤلفون آخرون: Takwa Bedhiafi (14153460) (author), Yousef Mohammad Hijji (14153463) (author), Nashiru Billa (4375261) (author)
منشور في: 2022
الموضوعات:
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author Sourour Idoudi (14153457)
author2 Takwa Bedhiafi (14153460)
Yousef Mohammad Hijji (14153463)
Nashiru Billa (4375261)
author2_role author
author
author
author_facet Sourour Idoudi (14153457)
Takwa Bedhiafi (14153460)
Yousef Mohammad Hijji (14153463)
Nashiru Billa (4375261)
author_role author
dc.creator.none.fl_str_mv Sourour Idoudi (14153457)
Takwa Bedhiafi (14153460)
Yousef Mohammad Hijji (14153463)
Nashiru Billa (4375261)
dc.date.none.fl_str_mv 2022-11-22T21:18:34Z
dc.identifier.none.fl_str_mv 10.1208/s12249-022-02268-y
dc.relation.none.fl_str_mv https://figshare.com/articles/journal_contribution/Curcumin_and_Derivatives_in_Nanoformulations_with_Therapeutic_Potential_on_Colorectal_Cancer/21598554
dc.rights.none.fl_str_mv CC BY 4.0
info:eu-repo/semantics/openAccess
dc.subject.none.fl_str_mv Pharmacology and pharmaceutical sciences
Drug Discovery
Pharmaceutical Science
Agronomy and Crop Science
Ecology
Aquatic Science
General Medicine
Ecology, Evolution, Behavior and Systematics
dc.title.none.fl_str_mv Curcumin and Derivatives in Nanoformulations with Therapeutic Potential on Colorectal Cancer
dc.type.none.fl_str_mv Text
Journal contribution
info:eu-repo/semantics/publishedVersion
text
contribution to journal
description <p>There is growing concern in the rise of colorectal cancer (CRC) cases globally, and with this rise is the presentation of drug resistance. Like other cancers, current treatment options are either invasive or manifest severe side effects. Thus, there is a move towards implementing safer treatment options. Curcumin (CUR), extracted from Curcuma longa, has received significant attention by scientists as possible alternative to chemotherapeutic agents. It is safe and effective against CRC and nontoxic in moderate concentrations. Crucially, it specifically modulates apoptotic effects on CRC. However, the use of CUR is limited by its low solubility and poor bioavailability in aqueous media. These limitations are surmountable through novel approaches, such as nanoencapsulation of CUR, which masks the physicochemical properties of CUR, thus potentiating its anti-CRC effects. Furthermore, chemical derivatization of CUR is another approach that can be used to address the above constraints. This review spans published work in the last two decades, with key findings employing either of the two approaches, in addition to a combined approach in managing CRC. The combined approach affords the possibility of better treatment outcomes but not widely investigated nor yet clinically implemented.</p> <p>Graphical Abstract</p><h2>Other Information</h2> <p> Published in: AAPS PharmSciTech<br> License: <a href="https://creativecommons.org/licenses/by/4.0" target="_blank">https://creativecommons.org/licenses/by/4.0</a><br>See article on publisher's website: <a href="http://dx.doi.org/10.1208/s12249-022-02268-y" target="_blank">http://dx.doi.org/10.1208/s12249-022-02268-y</a></p>
eu_rights_str_mv openAccess
id Manara2_7bfb5118646bfafef7a147bba9170a55
identifier_str_mv 10.1208/s12249-022-02268-y
network_acronym_str Manara2
network_name_str Manara2
oai_identifier_str oai:figshare.com:article/21598554
publishDate 2022
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rights_invalid_str_mv CC BY 4.0
spelling Curcumin and Derivatives in Nanoformulations with Therapeutic Potential on Colorectal CancerSourour Idoudi (14153457)Takwa Bedhiafi (14153460)Yousef Mohammad Hijji (14153463)Nashiru Billa (4375261)Pharmacology and pharmaceutical sciencesDrug DiscoveryPharmaceutical ScienceAgronomy and Crop ScienceEcologyAquatic ScienceGeneral MedicineEcology, Evolution, Behavior and Systematics<p>There is growing concern in the rise of colorectal cancer (CRC) cases globally, and with this rise is the presentation of drug resistance. Like other cancers, current treatment options are either invasive or manifest severe side effects. Thus, there is a move towards implementing safer treatment options. Curcumin (CUR), extracted from Curcuma longa, has received significant attention by scientists as possible alternative to chemotherapeutic agents. It is safe and effective against CRC and nontoxic in moderate concentrations. Crucially, it specifically modulates apoptotic effects on CRC. However, the use of CUR is limited by its low solubility and poor bioavailability in aqueous media. These limitations are surmountable through novel approaches, such as nanoencapsulation of CUR, which masks the physicochemical properties of CUR, thus potentiating its anti-CRC effects. Furthermore, chemical derivatization of CUR is another approach that can be used to address the above constraints. This review spans published work in the last two decades, with key findings employing either of the two approaches, in addition to a combined approach in managing CRC. The combined approach affords the possibility of better treatment outcomes but not widely investigated nor yet clinically implemented.</p> <p>Graphical Abstract</p><h2>Other Information</h2> <p> Published in: AAPS PharmSciTech<br> License: <a href="https://creativecommons.org/licenses/by/4.0" target="_blank">https://creativecommons.org/licenses/by/4.0</a><br>See article on publisher's website: <a href="http://dx.doi.org/10.1208/s12249-022-02268-y" target="_blank">http://dx.doi.org/10.1208/s12249-022-02268-y</a></p>2022-11-22T21:18:34ZTextJournal contributioninfo:eu-repo/semantics/publishedVersiontextcontribution to journal10.1208/s12249-022-02268-yhttps://figshare.com/articles/journal_contribution/Curcumin_and_Derivatives_in_Nanoformulations_with_Therapeutic_Potential_on_Colorectal_Cancer/21598554CC BY 4.0info:eu-repo/semantics/openAccessoai:figshare.com:article/215985542022-11-22T21:18:34Z
spellingShingle Curcumin and Derivatives in Nanoformulations with Therapeutic Potential on Colorectal Cancer
Sourour Idoudi (14153457)
Pharmacology and pharmaceutical sciences
Drug Discovery
Pharmaceutical Science
Agronomy and Crop Science
Ecology
Aquatic Science
General Medicine
Ecology, Evolution, Behavior and Systematics
status_str publishedVersion
title Curcumin and Derivatives in Nanoformulations with Therapeutic Potential on Colorectal Cancer
title_full Curcumin and Derivatives in Nanoformulations with Therapeutic Potential on Colorectal Cancer
title_fullStr Curcumin and Derivatives in Nanoformulations with Therapeutic Potential on Colorectal Cancer
title_full_unstemmed Curcumin and Derivatives in Nanoformulations with Therapeutic Potential on Colorectal Cancer
title_short Curcumin and Derivatives in Nanoformulations with Therapeutic Potential on Colorectal Cancer
title_sort Curcumin and Derivatives in Nanoformulations with Therapeutic Potential on Colorectal Cancer
topic Pharmacology and pharmaceutical sciences
Drug Discovery
Pharmaceutical Science
Agronomy and Crop Science
Ecology
Aquatic Science
General Medicine
Ecology, Evolution, Behavior and Systematics