The Effect of Exenatide on Cardiovascular Risk Markers in Women With Polycystic Ovary Syndrome

<h3>Background</h3><p dir="ltr">Polycystic ovary syndrome (PCOS) is associated with an adverse cardiovascular risk profile including a prothrombotic state. Exenatide has been shown to be effective at improving insulin sensitivity and weight loss in PCOS; therefore this st...

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التفاصيل البيبلوغرافية
المؤلف الرئيسي: Alison J. Dawson (18175003) (author)
مؤلفون آخرون: Thozhukat Sathyapalan (704787) (author), Rebecca Vince (17023392) (author), Anne-Marie Coady (18140278) (author), Ramzi A. Ajjan (3617486) (author), Eric S. Kilpatrick (6684365) (author), Stephen L. Atkin (6684368) (author)
منشور في: 2019
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author Alison J. Dawson (18175003)
author2 Thozhukat Sathyapalan (704787)
Rebecca Vince (17023392)
Anne-Marie Coady (18140278)
Ramzi A. Ajjan (3617486)
Eric S. Kilpatrick (6684365)
Stephen L. Atkin (6684368)
author2_role author
author
author
author
author
author
author_facet Alison J. Dawson (18175003)
Thozhukat Sathyapalan (704787)
Rebecca Vince (17023392)
Anne-Marie Coady (18140278)
Ramzi A. Ajjan (3617486)
Eric S. Kilpatrick (6684365)
Stephen L. Atkin (6684368)
author_role author
dc.creator.none.fl_str_mv Alison J. Dawson (18175003)
Thozhukat Sathyapalan (704787)
Rebecca Vince (17023392)
Anne-Marie Coady (18140278)
Ramzi A. Ajjan (3617486)
Eric S. Kilpatrick (6684365)
Stephen L. Atkin (6684368)
dc.date.none.fl_str_mv 2019-04-02T03:00:00Z
dc.identifier.none.fl_str_mv 10.3389/fendo.2019.00189
dc.relation.none.fl_str_mv https://figshare.com/articles/journal_contribution/The_Effect_of_Exenatide_on_Cardiovascular_Risk_Markers_in_Women_With_Polycystic_Ovary_Syndrome/25428340
dc.rights.none.fl_str_mv CC BY 4.0
info:eu-repo/semantics/openAccess
dc.subject.none.fl_str_mv Biomedical and clinical sciences
Clinical sciences
Reproductive medicine
polycystic ovary syndrome
exenatide
cardiovascular risk
endothelial function
inflammation
blood clot function
GLP-1 receptor agonists
dc.title.none.fl_str_mv The Effect of Exenatide on Cardiovascular Risk Markers in Women With Polycystic Ovary Syndrome
dc.type.none.fl_str_mv Text
Journal contribution
info:eu-repo/semantics/publishedVersion
text
contribution to journal
description <h3>Background</h3><p dir="ltr">Polycystic ovary syndrome (PCOS) is associated with an adverse cardiovascular risk profile including a prothrombotic state. Exenatide has been shown to be effective at improving insulin sensitivity and weight loss in PCOS; therefore this study was undertaken to assess its effects on weight, endothelial function, inflammatory markers, and fibrin structure/function in overweight/obese women with PCOS.</p><h3>Methods</h3><p dir="ltr">Thirty overweight/obese anovulatory women with all 3 Rotterdam criteria received exenatide 5 mcg bd for 4 weeks then 10 mcg bd for 12 weeks. The primary outcome was change in weight; secondary outcomes were changes in endothelial function [Reactive Hyperemia-Peripheral Arterial Tonometry (RH-PAT)], serum endothelial markers (ICAM-1, VCAM-1, E-selectin, and P-selectin), change in inflammation (hsCRP), and alteration in clot structure and function [maximum absorbance (MA), and time from full clot formation to 50% lysis (LT)].</p><h3>Results</h3><p dir="ltr">Twenty patients completed the study. Exenatide reduced weight 111.8 ± 4.8 to 108.6 ± 4.6 kg <i>p</i> = 0.003. Serum endothelial markers changed with a reduction in ICAM-1 (247.2 ± 12.9 to 231.3 ± 11.5 ng/ml <i>p</i> = 0.02), p-selectin (101.1 ± 8.2 to 87.4 ± 6.6 ng/ml <i>p</i> = 0.01), and e-selectin (38.5 ± 3.3 to 33.6 ± 2.6 ng/ml <i>p</i> = 0.03), without an overt change in endothelial function. Inflammation improved (CRP; 8.5 ± 1.4 to 5.6 ± 0.8 mmol/L <i>p</i> = 0.001), there was a reduction in clot function (LT; 2,987 ± 494 to 1,926 ± 321 s <i>p</i> = 0.02) but not clot structure.</p><h3>Conclusion</h3><p dir="ltr">Exenatide caused a 3% reduction in weight, improved serum markers of endothelial function, inflammation, and clot function reflecting an improvement in cardiovascular risk indices in these women with PCOS. This suggests exenatide could be an effective treatment for obese women with PCOS.</p><p dir="ltr">Clinical Trial Registration<b>:</b> ISRCTN81902209.</p><h2>Other Information</h2><p dir="ltr">Published in: Frontiers in Endocrinology<br>License: <a href="https://creativecommons.org/licenses/by/4.0/" target="_blank">https://creativecommons.org/licenses/by/4.0/</a><br>See article on publisher's website: <a href="https://dx.doi.org/10.3389/fendo.2019.00189" target="_blank">https://dx.doi.org/10.3389/fendo.2019.00189</a></p>
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identifier_str_mv 10.3389/fendo.2019.00189
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spelling The Effect of Exenatide on Cardiovascular Risk Markers in Women With Polycystic Ovary SyndromeAlison J. Dawson (18175003)Thozhukat Sathyapalan (704787)Rebecca Vince (17023392)Anne-Marie Coady (18140278)Ramzi A. Ajjan (3617486)Eric S. Kilpatrick (6684365)Stephen L. Atkin (6684368)Biomedical and clinical sciencesClinical sciencesReproductive medicinepolycystic ovary syndromeexenatidecardiovascular riskendothelial functioninflammationblood clot functionGLP-1 receptor agonists<h3>Background</h3><p dir="ltr">Polycystic ovary syndrome (PCOS) is associated with an adverse cardiovascular risk profile including a prothrombotic state. Exenatide has been shown to be effective at improving insulin sensitivity and weight loss in PCOS; therefore this study was undertaken to assess its effects on weight, endothelial function, inflammatory markers, and fibrin structure/function in overweight/obese women with PCOS.</p><h3>Methods</h3><p dir="ltr">Thirty overweight/obese anovulatory women with all 3 Rotterdam criteria received exenatide 5 mcg bd for 4 weeks then 10 mcg bd for 12 weeks. The primary outcome was change in weight; secondary outcomes were changes in endothelial function [Reactive Hyperemia-Peripheral Arterial Tonometry (RH-PAT)], serum endothelial markers (ICAM-1, VCAM-1, E-selectin, and P-selectin), change in inflammation (hsCRP), and alteration in clot structure and function [maximum absorbance (MA), and time from full clot formation to 50% lysis (LT)].</p><h3>Results</h3><p dir="ltr">Twenty patients completed the study. Exenatide reduced weight 111.8 ± 4.8 to 108.6 ± 4.6 kg <i>p</i> = 0.003. Serum endothelial markers changed with a reduction in ICAM-1 (247.2 ± 12.9 to 231.3 ± 11.5 ng/ml <i>p</i> = 0.02), p-selectin (101.1 ± 8.2 to 87.4 ± 6.6 ng/ml <i>p</i> = 0.01), and e-selectin (38.5 ± 3.3 to 33.6 ± 2.6 ng/ml <i>p</i> = 0.03), without an overt change in endothelial function. Inflammation improved (CRP; 8.5 ± 1.4 to 5.6 ± 0.8 mmol/L <i>p</i> = 0.001), there was a reduction in clot function (LT; 2,987 ± 494 to 1,926 ± 321 s <i>p</i> = 0.02) but not clot structure.</p><h3>Conclusion</h3><p dir="ltr">Exenatide caused a 3% reduction in weight, improved serum markers of endothelial function, inflammation, and clot function reflecting an improvement in cardiovascular risk indices in these women with PCOS. This suggests exenatide could be an effective treatment for obese women with PCOS.</p><p dir="ltr">Clinical Trial Registration<b>:</b> ISRCTN81902209.</p><h2>Other Information</h2><p dir="ltr">Published in: Frontiers in Endocrinology<br>License: <a href="https://creativecommons.org/licenses/by/4.0/" target="_blank">https://creativecommons.org/licenses/by/4.0/</a><br>See article on publisher's website: <a href="https://dx.doi.org/10.3389/fendo.2019.00189" target="_blank">https://dx.doi.org/10.3389/fendo.2019.00189</a></p>2019-04-02T03:00:00ZTextJournal contributioninfo:eu-repo/semantics/publishedVersiontextcontribution to journal10.3389/fendo.2019.00189https://figshare.com/articles/journal_contribution/The_Effect_of_Exenatide_on_Cardiovascular_Risk_Markers_in_Women_With_Polycystic_Ovary_Syndrome/25428340CC BY 4.0info:eu-repo/semantics/openAccessoai:figshare.com:article/254283402019-04-02T03:00:00Z
spellingShingle The Effect of Exenatide on Cardiovascular Risk Markers in Women With Polycystic Ovary Syndrome
Alison J. Dawson (18175003)
Biomedical and clinical sciences
Clinical sciences
Reproductive medicine
polycystic ovary syndrome
exenatide
cardiovascular risk
endothelial function
inflammation
blood clot function
GLP-1 receptor agonists
status_str publishedVersion
title The Effect of Exenatide on Cardiovascular Risk Markers in Women With Polycystic Ovary Syndrome
title_full The Effect of Exenatide on Cardiovascular Risk Markers in Women With Polycystic Ovary Syndrome
title_fullStr The Effect of Exenatide on Cardiovascular Risk Markers in Women With Polycystic Ovary Syndrome
title_full_unstemmed The Effect of Exenatide on Cardiovascular Risk Markers in Women With Polycystic Ovary Syndrome
title_short The Effect of Exenatide on Cardiovascular Risk Markers in Women With Polycystic Ovary Syndrome
title_sort The Effect of Exenatide on Cardiovascular Risk Markers in Women With Polycystic Ovary Syndrome
topic Biomedical and clinical sciences
Clinical sciences
Reproductive medicine
polycystic ovary syndrome
exenatide
cardiovascular risk
endothelial function
inflammation
blood clot function
GLP-1 receptor agonists