Image_1_Edonerpic maleate prevents epileptic seizure during recovery from brain damage by balancing excitatory and inhibitory inputs.TIF

<p>Functional recovery from brain damage, such as stroke, is a plastic process in the brain. The excitatory glutamate α-amino-3-hydroxy-5-methyl-4-isoxazole propionic acid receptor (AMPAR) plays a crucial role in neuronal functions, and the synaptic trafficking of AMPAR is a fundamental mechan...

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Main Author: Yuki Katsuno (20394911) (author)
Other Authors: Susumu Jitsuki (849442) (author), Wataru Ota (7372817) (author), Tomomi Yamanoue (20394914) (author), Hiroki Abe (1989742) (author), Takuya Takahashi (161915) (author)
Published: 2024
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_version_ 1852024636435333120
author Yuki Katsuno (20394911)
author2 Susumu Jitsuki (849442)
Wataru Ota (7372817)
Tomomi Yamanoue (20394914)
Hiroki Abe (1989742)
Takuya Takahashi (161915)
author2_role author
author
author
author
author
author_facet Yuki Katsuno (20394911)
Susumu Jitsuki (849442)
Wataru Ota (7372817)
Tomomi Yamanoue (20394914)
Hiroki Abe (1989742)
Takuya Takahashi (161915)
author_role author
dc.creator.none.fl_str_mv Yuki Katsuno (20394911)
Susumu Jitsuki (849442)
Wataru Ota (7372817)
Tomomi Yamanoue (20394914)
Hiroki Abe (1989742)
Takuya Takahashi (161915)
dc.date.none.fl_str_mv 2024-12-06T13:26:59Z
dc.identifier.none.fl_str_mv 10.3389/fncir.2024.1492043.s001
dc.relation.none.fl_str_mv https://figshare.com/articles/figure/Image_1_Edonerpic_maleate_prevents_epileptic_seizure_during_recovery_from_brain_damage_by_balancing_excitatory_and_inhibitory_inputs_TIF/27980492
dc.rights.none.fl_str_mv CC BY 4.0
info:eu-repo/semantics/openAccess
dc.subject.none.fl_str_mv Neuroscience
Central Nervous System
Neurocognitive Patterns and Neural Networks
Animal Neurobiology
AMPA receptors
edonerpic maleate
epileptic seizure
stroke
functional recovery
brain damage
synaptic plasticity
dc.title.none.fl_str_mv Image_1_Edonerpic maleate prevents epileptic seizure during recovery from brain damage by balancing excitatory and inhibitory inputs.TIF
dc.type.none.fl_str_mv Image
Figure
info:eu-repo/semantics/publishedVersion
image
description <p>Functional recovery from brain damage, such as stroke, is a plastic process in the brain. The excitatory glutamate α-amino-3-hydroxy-5-methyl-4-isoxazole propionic acid receptor (AMPAR) plays a crucial role in neuronal functions, and the synaptic trafficking of AMPAR is a fundamental mechanism underlying synaptic plasticity. We recently identified a collapsin response mediator protein 2 (CRMP2)-binding compound, edonerpic maleate, which augments rehabilitative training-dependent functional recovery from brain damage by facilitating experience-driven synaptic delivery of AMPARs. In animals recovering from cryogenic brain injury, a potential compensatory area adjacent to the injured region was observed, where the injection of CNQX, an AMPAR antagonist, significantly attenuated functional recovery. In the compensatory brain area of animals recovering from cryogenic injury, the administration of edonerpic maleate enhanced both excitatory and inhibitory synaptic inputs at pyramidal neurons. In contrast, recovered animals that did not receive the drug exhibited augmentation of only excitatory synaptic input. The threshold of picrotoxin-induced epileptic seizure in recovered animals without edonerpic maleate treatment was lower than in intact animals and recovered animals with edonerpic maleate. Thus, edonerpic maleate enhances motor function recovery from brain damage by balancing excitatory and inhibitory synaptic inputs, which helps prevent epileptic seizures during recovery.</p>
eu_rights_str_mv openAccess
id Manara_977cd2bb9bd2d2d09928dc50ffdcaff2
identifier_str_mv 10.3389/fncir.2024.1492043.s001
network_acronym_str Manara
network_name_str ManaraRepo
oai_identifier_str oai:figshare.com:article/27980492
publishDate 2024
repository.mail.fl_str_mv
repository.name.fl_str_mv
repository_id_str
rights_invalid_str_mv CC BY 4.0
spelling Image_1_Edonerpic maleate prevents epileptic seizure during recovery from brain damage by balancing excitatory and inhibitory inputs.TIFYuki Katsuno (20394911)Susumu Jitsuki (849442)Wataru Ota (7372817)Tomomi Yamanoue (20394914)Hiroki Abe (1989742)Takuya Takahashi (161915)NeuroscienceCentral Nervous SystemNeurocognitive Patterns and Neural NetworksAnimal NeurobiologyAMPA receptorsedonerpic maleateepileptic seizurestrokefunctional recoverybrain damagesynaptic plasticity<p>Functional recovery from brain damage, such as stroke, is a plastic process in the brain. The excitatory glutamate α-amino-3-hydroxy-5-methyl-4-isoxazole propionic acid receptor (AMPAR) plays a crucial role in neuronal functions, and the synaptic trafficking of AMPAR is a fundamental mechanism underlying synaptic plasticity. We recently identified a collapsin response mediator protein 2 (CRMP2)-binding compound, edonerpic maleate, which augments rehabilitative training-dependent functional recovery from brain damage by facilitating experience-driven synaptic delivery of AMPARs. In animals recovering from cryogenic brain injury, a potential compensatory area adjacent to the injured region was observed, where the injection of CNQX, an AMPAR antagonist, significantly attenuated functional recovery. In the compensatory brain area of animals recovering from cryogenic injury, the administration of edonerpic maleate enhanced both excitatory and inhibitory synaptic inputs at pyramidal neurons. In contrast, recovered animals that did not receive the drug exhibited augmentation of only excitatory synaptic input. The threshold of picrotoxin-induced epileptic seizure in recovered animals without edonerpic maleate treatment was lower than in intact animals and recovered animals with edonerpic maleate. Thus, edonerpic maleate enhances motor function recovery from brain damage by balancing excitatory and inhibitory synaptic inputs, which helps prevent epileptic seizures during recovery.</p>2024-12-06T13:26:59ZImageFigureinfo:eu-repo/semantics/publishedVersionimage10.3389/fncir.2024.1492043.s001https://figshare.com/articles/figure/Image_1_Edonerpic_maleate_prevents_epileptic_seizure_during_recovery_from_brain_damage_by_balancing_excitatory_and_inhibitory_inputs_TIF/27980492CC BY 4.0info:eu-repo/semantics/openAccessoai:figshare.com:article/279804922024-12-06T13:26:59Z
spellingShingle Image_1_Edonerpic maleate prevents epileptic seizure during recovery from brain damage by balancing excitatory and inhibitory inputs.TIF
Yuki Katsuno (20394911)
Neuroscience
Central Nervous System
Neurocognitive Patterns and Neural Networks
Animal Neurobiology
AMPA receptors
edonerpic maleate
epileptic seizure
stroke
functional recovery
brain damage
synaptic plasticity
status_str publishedVersion
title Image_1_Edonerpic maleate prevents epileptic seizure during recovery from brain damage by balancing excitatory and inhibitory inputs.TIF
title_full Image_1_Edonerpic maleate prevents epileptic seizure during recovery from brain damage by balancing excitatory and inhibitory inputs.TIF
title_fullStr Image_1_Edonerpic maleate prevents epileptic seizure during recovery from brain damage by balancing excitatory and inhibitory inputs.TIF
title_full_unstemmed Image_1_Edonerpic maleate prevents epileptic seizure during recovery from brain damage by balancing excitatory and inhibitory inputs.TIF
title_short Image_1_Edonerpic maleate prevents epileptic seizure during recovery from brain damage by balancing excitatory and inhibitory inputs.TIF
title_sort Image_1_Edonerpic maleate prevents epileptic seizure during recovery from brain damage by balancing excitatory and inhibitory inputs.TIF
topic Neuroscience
Central Nervous System
Neurocognitive Patterns and Neural Networks
Animal Neurobiology
AMPA receptors
edonerpic maleate
epileptic seizure
stroke
functional recovery
brain damage
synaptic plasticity