Bitopic Sigma 1 Receptor Modulators to Shed Light on Molecular Mechanisms Underpinning Ligand Binding and Receptor Oligomerization

The sigma 1 receptor (S1R) is an enigmatic ligand-operated chaperone involved in many important biological processes, and its functions are not fully understood yet. Herein, we developed a novel series of bitopic S1R ligands as versatile tools to investigate binding processes, allosteric modulation,...

Full description

Saved in:
Bibliographic Details
Main Author: Giacomo Rossino (8162412) (author)
Other Authors: Marta Rui (6694853) (author), Pasquale Linciano (4426435) (author), Daniela Rossi (1716643) (author), Massimo Boiocchi (1497415) (author), Marco Peviani (517091) (author), Elena Poggio (11540406) (author), Daniela Curti (2339923) (author), Dirk Schepmann (1484284) (author), Bernhard Wünsch (1484308) (author), Mariela González-Avendaño (8162418) (author), Ariela Vergara-Jaque (638616) (author), Julio Caballero (531146) (author), Simona Collina (136811) (author)
Published: 2021
Subjects:
Tags: Add Tag
No Tags, Be the first to tag this record!