Kinetics of ultrasonic release of doxorubicin from pluronic P105 micelles

The aim of this research was to measure and model the kinetics of acoustic release and subsequent re-encapsulation of Doxorubicin (DOX) from Pluronic P105 micelles. A fluorescence detection ultrasound exposure chamber was used. Experimental data showed that no significant release was observed when D...

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Main Author: Husseini, Ghaleb (author)
Other Authors: Rapoport, Natalya Y. (author), Christensen, Douglas A. (author), Pruitt, John D. (author), Pitt, William G. (author)
Format: article
Published: 2001
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Online Access:http://hdl.handle.net/11073/19830
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author Husseini, Ghaleb
author2 Rapoport, Natalya Y.
Christensen, Douglas A.
Pruitt, John D.
Pitt, William G.
author2_role author
author
author
author
author_facet Husseini, Ghaleb
Rapoport, Natalya Y.
Christensen, Douglas A.
Pruitt, John D.
Pitt, William G.
author_role author
dc.creator.none.fl_str_mv Husseini, Ghaleb
Rapoport, Natalya Y.
Christensen, Douglas A.
Pruitt, John D.
Pitt, William G.
dc.date.none.fl_str_mv 2001
2020-12-21T05:06:37Z
2020-12-21T05:06:37Z
dc.format.none.fl_str_mv application/pdf
dc.identifier.none.fl_str_mv Husseini, G. A., Rapoport, N. Y., Christensen, D. A., Pruitt, J. D., & Pitt, W. G. (2002). Kinetics of ultrasonic release of doxorubicin from pluronic P105 micelles. Colloids and Surfaces B: Biointerfaces, 24(3–4), 253–264. https://doi.org/10.1016/s0927-7765(01)00273-9
0927-7765
http://hdl.handle.net/11073/19830
10.1016/s0927-7765(01)00273-9
dc.language.none.fl_str_mv en_US
dc.publisher.none.fl_str_mv Elsevier
dc.relation.none.fl_str_mv https://doi.org/10.1016/s0927-7765(01)00273-9
dc.subject.none.fl_str_mv Micellar drug delivery
Doxorubicin
Pulsed ultrasound
Fluorescence measurement
Kinetic models
dc.title.none.fl_str_mv Kinetics of ultrasonic release of doxorubicin from pluronic P105 micelles
dc.type.none.fl_str_mv Peer-Reviewed
Postprint
info:eu-repo/semantics/publishedVersion
info:eu-repo/semantics/article
description The aim of this research was to measure and model the kinetics of acoustic release and subsequent re-encapsulation of Doxorubicin (DOX) from Pluronic P105 micelles. A fluorescence detection ultrasound exposure chamber was used. Experimental data showed that no significant release was observed when DOX loaded in Pluronic P105 micelles was exposed to ultrasound for less than 0.1 s at a power density of 58 mW/cm2 and a frequency of 20 kHz. Above this threshold, the amount of release was shown to increase as the pulse length increased up to 0.6 s. The same experiments showed that it requires at least 0.1 s of no ultrasound for measurable re-encapsulation to occur. Release and re-encapsulation are completed within about 0.6 s of the beginning of the ON and OFF phases of pulsed ultrasound. Several physical models and their corresponding mathematical solutions were analyzed to see which most closely fit the data. The model of zero-order release with first-order re-encapsulation appears to represent data from this polymeric system better than other models. This technique has possible applications in site-specific chemotherapy.
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identifier_str_mv Husseini, G. A., Rapoport, N. Y., Christensen, D. A., Pruitt, J. D., & Pitt, W. G. (2002). Kinetics of ultrasonic release of doxorubicin from pluronic P105 micelles. Colloids and Surfaces B: Biointerfaces, 24(3–4), 253–264. https://doi.org/10.1016/s0927-7765(01)00273-9
0927-7765
10.1016/s0927-7765(01)00273-9
language_invalid_str_mv en_US
network_acronym_str aus
network_name_str aus
oai_identifier_str oai:repository.aus.edu:11073/19830
publishDate 2001
publisher.none.fl_str_mv Elsevier
repository.mail.fl_str_mv
repository.name.fl_str_mv
repository_id_str
spelling Kinetics of ultrasonic release of doxorubicin from pluronic P105 micellesHusseini, GhalebRapoport, Natalya Y.Christensen, Douglas A.Pruitt, John D.Pitt, William G.Micellar drug deliveryDoxorubicinPulsed ultrasoundFluorescence measurementKinetic modelsThe aim of this research was to measure and model the kinetics of acoustic release and subsequent re-encapsulation of Doxorubicin (DOX) from Pluronic P105 micelles. A fluorescence detection ultrasound exposure chamber was used. Experimental data showed that no significant release was observed when DOX loaded in Pluronic P105 micelles was exposed to ultrasound for less than 0.1 s at a power density of 58 mW/cm2 and a frequency of 20 kHz. Above this threshold, the amount of release was shown to increase as the pulse length increased up to 0.6 s. The same experiments showed that it requires at least 0.1 s of no ultrasound for measurable re-encapsulation to occur. Release and re-encapsulation are completed within about 0.6 s of the beginning of the ON and OFF phases of pulsed ultrasound. Several physical models and their corresponding mathematical solutions were analyzed to see which most closely fit the data. The model of zero-order release with first-order re-encapsulation appears to represent data from this polymeric system better than other models. This technique has possible applications in site-specific chemotherapy.Elsevier2020-12-21T05:06:37Z2020-12-21T05:06:37Z2001Peer-ReviewedPostprintinfo:eu-repo/semantics/publishedVersioninfo:eu-repo/semantics/articleapplication/pdfHusseini, G. A., Rapoport, N. Y., Christensen, D. A., Pruitt, J. D., & Pitt, W. G. (2002). Kinetics of ultrasonic release of doxorubicin from pluronic P105 micelles. Colloids and Surfaces B: Biointerfaces, 24(3–4), 253–264. https://doi.org/10.1016/s0927-7765(01)00273-90927-7765http://hdl.handle.net/11073/1983010.1016/s0927-7765(01)00273-9en_UShttps://doi.org/10.1016/s0927-7765(01)00273-9oai:repository.aus.edu:11073/198302024-08-22T12:04:46Z
spellingShingle Kinetics of ultrasonic release of doxorubicin from pluronic P105 micelles
Husseini, Ghaleb
Micellar drug delivery
Doxorubicin
Pulsed ultrasound
Fluorescence measurement
Kinetic models
status_str publishedVersion
title Kinetics of ultrasonic release of doxorubicin from pluronic P105 micelles
title_full Kinetics of ultrasonic release of doxorubicin from pluronic P105 micelles
title_fullStr Kinetics of ultrasonic release of doxorubicin from pluronic P105 micelles
title_full_unstemmed Kinetics of ultrasonic release of doxorubicin from pluronic P105 micelles
title_short Kinetics of ultrasonic release of doxorubicin from pluronic P105 micelles
title_sort Kinetics of ultrasonic release of doxorubicin from pluronic P105 micelles
topic Micellar drug delivery
Doxorubicin
Pulsed ultrasound
Fluorescence measurement
Kinetic models
url http://hdl.handle.net/11073/19830