DNA damage induced by micellar-delivered doxorubicin and ultrasound: comet assay study

To minimize adverse side effects of chemotherapy, we have developed a micellar drug carrier that retains hydrophobic drugs, and then releases the drug by ultrasonic stimulation. This study investigated the DNA damage induced by doxorubicin (DOX) delivered to human leukemia (HL-60) cells from pluroni...

وصف كامل

محفوظ في:
التفاصيل البيبلوغرافية
المؤلف الرئيسي: Husseini, Ghaleb (author)
مؤلفون آخرون: El-Fayoumi, Refaat I. (author), O'Neill, Kim L. (author), Rapoport, Natalya Y. (author), Pitt, William G. (author)
التنسيق: article
منشور في: 2000
الموضوعات:
الوصول للمادة أونلاين:http://hdl.handle.net/11073/19827
الوسوم: إضافة وسم
لا توجد وسوم, كن أول من يضع وسما على هذه التسجيلة!
_version_ 1864513440240893952
author Husseini, Ghaleb
author2 El-Fayoumi, Refaat I.
O'Neill, Kim L.
Rapoport, Natalya Y.
Pitt, William G.
author2_role author
author
author
author
author_facet Husseini, Ghaleb
El-Fayoumi, Refaat I.
O'Neill, Kim L.
Rapoport, Natalya Y.
Pitt, William G.
author_role author
dc.creator.none.fl_str_mv Husseini, Ghaleb
El-Fayoumi, Refaat I.
O'Neill, Kim L.
Rapoport, Natalya Y.
Pitt, William G.
dc.date.none.fl_str_mv 2000
2020-12-17T05:08:26Z
2020-12-17T05:08:26Z
dc.format.none.fl_str_mv application/pdf
dc.identifier.none.fl_str_mv Husseini, G. A., El-Fayoumi, R. I., O’Neill, K. L., Rapoport, N. Y., & Pitt, W. G. (2000). DNA damage induced by micellar-delivered doxorubicin and ultrasound: comet assay study. Cancer Letters, 154(2), 211–216. https://doi.org/10.1016/s0304-3835(00)00399-2
0304-3835
http://hdl.handle.net/11073/19827
10.1016/S0304-3835(00)00399-2
dc.language.none.fl_str_mv en_US
dc.publisher.none.fl_str_mv Elsevier
dc.relation.none.fl_str_mv https://doi.org/10.1016/S0304-3835(00)00399-2
dc.subject.none.fl_str_mv Micellar drug delivery
Doxorubicin
Comet assay
Ultrasound
dc.title.none.fl_str_mv DNA damage induced by micellar-delivered doxorubicin and ultrasound: comet assay study
dc.type.none.fl_str_mv Peer-Reviewed
Postprint
info:eu-repo/semantics/publishedVersion
info:eu-repo/semantics/article
description To minimize adverse side effects of chemotherapy, we have developed a micellar drug carrier that retains hydrophobic drugs, and then releases the drug by ultrasonic stimulation. This study investigated the DNA damage induced by doxorubicin (DOX) delivered to human leukemia (HL-60) cells from pluronic P-105 micelles with and without the application of ultrasound. The comet assay was used to quantify the amount of DNA damage. No significant DNA damage was observed when the cells were treated with 0.1, 1 and 10 wt% P-105 with or without ultrasound (70 kHz, 1.3 W/cm2) for 1 h or for up to 3 h in 10 wt% P-105. However, when cells were incubated with 10 μg/ml free DOX for up to 9 h, DNA damage increased with incubation time (P=0.0011). Exposure of cells to the same concentration of DOX in the presence of 10-wt% P-105 showed no significant DNA damage for up to 9 h of incubation. However, when ultrasound was applied, a rapid and significant increase in DNA damage was observed (P=0.0001). The application of ultrasound causes the release of DOX from micelles or causes the HL-60 cells to take up the micelle encapsulated DOX. Our experiments indicated that the combination of DOX, ultrasound and pluronic P105 causes the largest DNA damage to HL-60 cells. We believe that this technique can be used for controlled drug delivery.
format article
id aus_cfc2c582a634369d915b8bd5904d9ad6
identifier_str_mv Husseini, G. A., El-Fayoumi, R. I., O’Neill, K. L., Rapoport, N. Y., & Pitt, W. G. (2000). DNA damage induced by micellar-delivered doxorubicin and ultrasound: comet assay study. Cancer Letters, 154(2), 211–216. https://doi.org/10.1016/s0304-3835(00)00399-2
0304-3835
10.1016/S0304-3835(00)00399-2
language_invalid_str_mv en_US
network_acronym_str aus
network_name_str aus
oai_identifier_str oai:repository.aus.edu:11073/19827
publishDate 2000
publisher.none.fl_str_mv Elsevier
repository.mail.fl_str_mv
repository.name.fl_str_mv
repository_id_str
spelling DNA damage induced by micellar-delivered doxorubicin and ultrasound: comet assay studyHusseini, GhalebEl-Fayoumi, Refaat I.O'Neill, Kim L.Rapoport, Natalya Y.Pitt, William G.Micellar drug deliveryDoxorubicinComet assayUltrasoundTo minimize adverse side effects of chemotherapy, we have developed a micellar drug carrier that retains hydrophobic drugs, and then releases the drug by ultrasonic stimulation. This study investigated the DNA damage induced by doxorubicin (DOX) delivered to human leukemia (HL-60) cells from pluronic P-105 micelles with and without the application of ultrasound. The comet assay was used to quantify the amount of DNA damage. No significant DNA damage was observed when the cells were treated with 0.1, 1 and 10 wt% P-105 with or without ultrasound (70 kHz, 1.3 W/cm2) for 1 h or for up to 3 h in 10 wt% P-105. However, when cells were incubated with 10 μg/ml free DOX for up to 9 h, DNA damage increased with incubation time (P=0.0011). Exposure of cells to the same concentration of DOX in the presence of 10-wt% P-105 showed no significant DNA damage for up to 9 h of incubation. However, when ultrasound was applied, a rapid and significant increase in DNA damage was observed (P=0.0001). The application of ultrasound causes the release of DOX from micelles or causes the HL-60 cells to take up the micelle encapsulated DOX. Our experiments indicated that the combination of DOX, ultrasound and pluronic P105 causes the largest DNA damage to HL-60 cells. We believe that this technique can be used for controlled drug delivery.Elsevier2020-12-17T05:08:26Z2020-12-17T05:08:26Z2000Peer-ReviewedPostprintinfo:eu-repo/semantics/publishedVersioninfo:eu-repo/semantics/articleapplication/pdfHusseini, G. A., El-Fayoumi, R. I., O’Neill, K. L., Rapoport, N. Y., & Pitt, W. G. (2000). DNA damage induced by micellar-delivered doxorubicin and ultrasound: comet assay study. Cancer Letters, 154(2), 211–216. https://doi.org/10.1016/s0304-3835(00)00399-20304-3835http://hdl.handle.net/11073/1982710.1016/S0304-3835(00)00399-2en_UShttps://doi.org/10.1016/S0304-3835(00)00399-2oai:repository.aus.edu:11073/198272024-08-22T12:04:27Z
spellingShingle DNA damage induced by micellar-delivered doxorubicin and ultrasound: comet assay study
Husseini, Ghaleb
Micellar drug delivery
Doxorubicin
Comet assay
Ultrasound
status_str publishedVersion
title DNA damage induced by micellar-delivered doxorubicin and ultrasound: comet assay study
title_full DNA damage induced by micellar-delivered doxorubicin and ultrasound: comet assay study
title_fullStr DNA damage induced by micellar-delivered doxorubicin and ultrasound: comet assay study
title_full_unstemmed DNA damage induced by micellar-delivered doxorubicin and ultrasound: comet assay study
title_short DNA damage induced by micellar-delivered doxorubicin and ultrasound: comet assay study
title_sort DNA damage induced by micellar-delivered doxorubicin and ultrasound: comet assay study
topic Micellar drug delivery
Doxorubicin
Comet assay
Ultrasound
url http://hdl.handle.net/11073/19827