The molecular mechanisms of plasticity in crystal forms of theophylline

Plastic and elastic behaviors of organic crystals have profound influence on the processability of pharmaceutical substances. Analogous to metals, the identifications of molecular slip planes in organic crystals are regarded as a strategy for harnessing plasticity. In this work, we experimentally ch...

وصف كامل

محفوظ في:
التفاصيل البيبلوغرافية
المؤلف الرئيسي: Liu, Hongji (author)
مؤلفون آخرون: Chan, H.C. Stephen (author), Zhang, Li (author), Lu, Yang (author), Li, Jiaquan (author), Li, Jianting (author), Li, Liang (author), Zhou, Zhengzheng (author)
منشور في: 2023
الموضوعات:
الوصول للمادة أونلاين:https://depot.sorbonne.ae/handle/20.500.12458/1622
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author Liu, Hongji
author2 Chan, H.C. Stephen
Zhang, Li
Lu, Yang
Li, Jiaquan
Li, Jianting
Li, Liang
Zhou, Zhengzheng
author2_role author
author
author
author
author
author
author
author_facet Liu, Hongji
Chan, H.C. Stephen
Zhang, Li
Lu, Yang
Li, Jiaquan
Li, Jianting
Li, Liang
Zhou, Zhengzheng
author_role author
dc.creator.none.fl_str_mv Liu, Hongji
Chan, H.C. Stephen
Zhang, Li
Lu, Yang
Li, Jiaquan
Li, Jianting
Li, Liang
Zhou, Zhengzheng
dc.date.none.fl_str_mv 2023
2024-06-24T11:56:43Z
2024-06-24T11:56:43Z
dc.identifier.none.fl_str_mv 1001-8417
https://depot.sorbonne.ae/handle/20.500.12458/1622
10.1016/j.cclet.2022.108057
dc.language.none.fl_str_mv en
dc.relation.none.fl_str_mv Chinese Chemical Letters
dc.subject.none.fl_str_mv Theophylline
Elasticity
Plastic crystal
Density functional theory
Mechanochemistry
dc.title.none.fl_str_mv The molecular mechanisms of plasticity in crystal forms of theophylline
dc.type.none.fl_str_mv Controlled Vocabulary for Resource Type Genres::text::periodical::journal::contribution to journal::journal article
description Plastic and elastic behaviors of organic crystals have profound influence on the processability of pharmaceutical substances. Analogous to metals, the identifications of molecular slip planes in organic crystals are regarded as a strategy for harnessing plasticity. In this work, we experimentally characterized the form II anhydrous theophylline (THPa) and its monohydrate (THPm) for their distinct plastic and elastic behaviors. Extensive DFT calculations were performed to model the effects of increasing lattice strains on molecular packing. We discovered that the energy barrier associated with the strain-induced molecular rearrangement would link to the plasticity of THPa, and possibly other simple aromatic compounds. Meanwhile, water molecules in THPm disrupt the stacking architecture from THPm and effectively undermine the general mechanism for plasticity. Hydrate formation would therefore be an alternative strategy to engineer the mechanical property of organic crystalline materials.
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identifier_str_mv 1001-8417
10.1016/j.cclet.2022.108057
language_invalid_str_mv en
network_acronym_str sorbonner
network_name_str Sorbonne University Abu Dhabi repository
oai_identifier_str oai:depot.sorbonne.ae:20.500.12458/1622
publishDate 2023
repository.mail.fl_str_mv
repository.name.fl_str_mv
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spelling The molecular mechanisms of plasticity in crystal forms of theophyllineLiu, HongjiChan, H.C. StephenZhang, LiLu, YangLi, JiaquanLi, JiantingLi, LiangZhou, ZhengzhengTheophyllineElasticityPlastic crystalDensity functional theoryMechanochemistryPlastic and elastic behaviors of organic crystals have profound influence on the processability of pharmaceutical substances. Analogous to metals, the identifications of molecular slip planes in organic crystals are regarded as a strategy for harnessing plasticity. In this work, we experimentally characterized the form II anhydrous theophylline (THPa) and its monohydrate (THPm) for their distinct plastic and elastic behaviors. Extensive DFT calculations were performed to model the effects of increasing lattice strains on molecular packing. We discovered that the energy barrier associated with the strain-induced molecular rearrangement would link to the plasticity of THPa, and possibly other simple aromatic compounds. Meanwhile, water molecules in THPm disrupt the stacking architecture from THPm and effectively undermine the general mechanism for plasticity. Hydrate formation would therefore be an alternative strategy to engineer the mechanical property of organic crystalline materials.2024-06-24T11:56:43Z2024-06-24T11:56:43Z2023Controlled Vocabulary for Resource Type Genres::text::periodical::journal::contribution to journal::journal article1001-8417https://depot.sorbonne.ae/handle/20.500.12458/162210.1016/j.cclet.2022.108057enChinese Chemical Lettersoai:depot.sorbonne.ae:20.500.12458/16222024-06-24T11:56:43Z
spellingShingle The molecular mechanisms of plasticity in crystal forms of theophylline
Liu, Hongji
Theophylline
Elasticity
Plastic crystal
Density functional theory
Mechanochemistry
title The molecular mechanisms of plasticity in crystal forms of theophylline
title_full The molecular mechanisms of plasticity in crystal forms of theophylline
title_fullStr The molecular mechanisms of plasticity in crystal forms of theophylline
title_full_unstemmed The molecular mechanisms of plasticity in crystal forms of theophylline
title_short The molecular mechanisms of plasticity in crystal forms of theophylline
title_sort The molecular mechanisms of plasticity in crystal forms of theophylline
topic Theophylline
Elasticity
Plastic crystal
Density functional theory
Mechanochemistry
url https://depot.sorbonne.ae/handle/20.500.12458/1622